Synthesis and antibacterial activity of some pyrazol-1-ylquinoxalin-2(1H)-one derivatives

Synthesis and antibacterial activity of some pyrazol-1-ylquinoxalin-2(1H)-one derivatives

3-Hydrazinoquinoxalin-2(1H)-one was prepared from quinoxaline-2,3-dione and subsequently used for the synthesis of some potentially biologically active 3-(pyrazol-1-yl)quinoxalin-2(1H)-one derivatives. While 3-(3,5-dimethylpyrazol-1-yl)quinoxalin-2(1H)-one showed a comparative effect with streptomycin, 3-(5-oxo-3-phenyl-4,5-di- hydropyrazol-1-yl)quinoxalin-2(1H)-one was found to be the most...
 
Published at Chemistry of Heterocyclic Compounds
Volume 45
Issue 11
Pages 1370-1378
Published in 2009
 
 
visit (http://link.springer.com/journal/10593/45/11/page/1)
 
 
Ajani, O.O., Obafemi C.A., Ikpo, C.O., Ogunniran K.O. and Nwinyi, O.C.
AJANI OLAYINKA OYEWALE » Prof. Olayinka Oyewale AJANI is an expeditious chemist who has distinguished himself both as a seasoned industrialist and a prolific researcher in the academic world especially in the area of Organic Synthesis and Medicinal Chemistry. He obtained his Master’s degree in Chemistry in 2006 from Obafemi Awolowo University, Ile-ife, Osun State, Nigeria. In 2012, Ajani O.O. obtained his Doctoral... view full profile
AJANI OLAYINKA OYEWALE
 
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