Microwave assisted synthesis and evaluation of antimicrobial activity of 3-{3-(s-aryl and s-heteroaromatic) acryloyl}-2H-chromen-2-one derivatives

Microwave assisted synthesis and evaluation of antimicrobial activity of 3-{3-(s-aryl and s-heteroaromatic) acryloyl}-2H-chromen-2-one derivatives

The exploration of potential utilization of microwaves as an energy source for heterocyclic synthesis was herein investigated using condensation of 3-acetylcoumarin (1) with aromatic and heteroaromatic aldehydes to afford the corresponding aromatic chalcones (2a–j) and heteroaromatic chalcones (3a–e and 4a–e), respectively, in good to excellent yield within 1–3 min. The chemical...
 
Published at Journal of Heterocyclic Chemistry
Volume 47
Issue 1
Pages 179-187
Published in 2010
 
 
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Ajani, O.O. and Nwinyi, O.C.
AJANI OLAYINKA OYEWALE » Prof. Olayinka Oyewale AJANI is an expeditious chemist who has distinguished himself both as a seasoned industrialist and a prolific researcher in the academic world especially in the area of Organic Synthesis and Medicinal Chemistry. He obtained his Master’s degree in Chemistry in 2006 from Obafemi Awolowo University, Ile-ife, Osun State, Nigeria. In 2012, Ajani O.O. obtained his Doctoral... view full profile
AJANI OLAYINKA OYEWALE
 
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