Facile Synthesis and Characterization of New 2,3-Disubstituted Benzimidazole Derivatives

Facile Synthesis and Characterization of New 2,3-Disubstituted Benzimidazole Derivatives

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Benzimidazoles are known to represent a class of medicinally important compounds which are extensively used as antibacterial agents. Hence, a series of five 2-substitutedbenzimidazole precursors (1a-e) were synthesized via [4 + 1] condensation and imino compound (1f) by simple condensation in the presence of Conc. HCl as catalyst. Synthetic modification of N-1 position was achieved in order to...
 
Published at International Research Journal of Pure and Applied Chemistry
Volume 3
Issue 1
Pages 10-21
 
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Ajani, O.O., Ezeoke E.K., Edobor-Osoh, A. and Ajani, A.O.
AJANI OLAYINKA OYEWALE » Prof. Olayinka Oyewale AJANI is an expeditious chemist who has distinguished himself both as a seasoned industrialist and a prolific researcher in the academic world especially in the area of Organic Synthesis and Medicinal Chemistry. He obtained his Master’s degree in Chemistry in 2006 from Obafemi Awolowo University, Ile-ife, Osun State, Nigeria. In 2012, Ajani O.O. obtained his Doctoral... view full profile
AJANI OLAYINKA OYEWALE
 
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